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Wiley电子期刊(11)	ProQuest学位论文(1)	Elsevier电子期刊(1572)
SpringerLink电子期刊(552)	NATURE电子期刊(12)	ACS电子期刊(248)

在“Elsevier电子期刊”中，命中：1,572条，耗时：0.0829584 秒

在所有数据库中总计命中：2,396条

1.Inhibition kinetics and molecular simulation of p-substituted cinnamic acid derivatives on tyrosinase

作者：Yi Cui^a ; Yong-Hua Hu^a ; Feng Yu^a ; Jing Zheng^a ; Lin-Shan Chen^a ; Qing-Xi Chen^a ; ^b ; Qin Wang^a ; ^{qwang@xmu.edu.cn}

关键词：4-CCA ; 4-chlorocinnamic acid ; 4-ECA ; 4-ethoxycinnamic acid ; 4-NCA ; 4-nitrocinnamic acid ; DMSO ; dimethyl-sulfoxide ; L-Tyr ; L-tyrosine ; L-DOPA ; L-3 ; 4-Dihydroxyphenylalanine ; Km ; Michaelis-Menten constant ; KI ; equilibrium constant of the inhibitor combining with the free enzyme ; IC50 ; inhibitor concentration leading to a 50% loss of activity

刊名：International Journal of Biological Macromolecules

出版年：2017

2.A new set of assays for the discovery of aminoacyl-tRNA synthetase inhibitors

作者：Adé ; laï ; de Saint-Lé ; ger^a ; Lluí ; s Ribas de Pouplana^a ; ^b ; ^c ; ^{lluis.ribas@irbbarcelona.org}

关键词：ARS ; aminoacyl-tRNA synthetases ; Cpd ; compound ; HTS ; high throughput screening ; IC50 ; half maximal inhibitory concentration ; Km ; Michaelis constant ; LRS ; leucyl-tRNA synthetase ; MIC ; minimum inhibitory concentration ; OM ; Omnia Molecular ; RLU ; relative light unit ; RRS ; arginyl-tRNA synthetase ; RT ; room temperature ; SRS ; seryl-tRNA synthetase ; SD ; standard deviation ; tRNA ; aminoacylate transfer RNA ; YRS ; tyrosyl-tRNA synthetase ; WRS ; tryptophanyl-tRNA synthetase ; Wt ; wild-type

刊名：Methods

出版年：2017

3.Combining in silico and in vitro approaches to evaluate the acetylcholinesterase inhibitory profile of some commercially available flavonoids in the management of Alzheimer’s disease

作者：Asokkumar Kuppusamy^a ; Madeswaran Arumugam^a ; ^{madeswaran2@gmail.com} ; Sonia George^b

关键词：Alzheimer&rsquo ; s disease ; Binding energy ; Inhibition constant ; Amino acid residues ; Molecular interactions

刊名：International Journal of Biological Macromolecules

出版年：2017

4.Chiral resolution of serial potent and selective σ₁ ligands and biological evaluation of (−)-[¹⁸F]TZ3108 in rodent and the nonhuman primate brain

作者：Xuyi Yue^a ; Hongjun Jin^a ; Zonghua Luo^a ; Hui Liu^a ; Xiang Zhang^a ; Ethan D. McSpadden^b ; Linlin Tian^c ; Hubert P. Flores^c ; Joel S. Perlmutter^a ; ^c ; Stanley M. Parsons^b ; Zhude Tu^a ; ^{tuz@mir.wustl.edu}

关键词：calcd ; calculated ; CH2Cl2 ; dichloromethane ; CNS ; central nervous system ; DMSO ; dimethyl sulfoxide ; [3H]DTG ; [3H]ditolylguanidine ; DTTA ; di-p-toluoyl tartaric acid ; EBP ; emopamil binding protein ; ee ; enantiomeric excess ; EOB ; end of bombardment ; EtOH ; ethanol ; [18F]FTC146 ; 18F-6-(3-fluoropropyl)-3-(2-(azepan-1-yl)ethyl)benzo[d]thiazol-2(3H)-one ; HPLC ; high performance liquid chromatography ; HRMS ; high resolution mass spectrometry ; IC50 ; half maximum inhibitory constant ; K2CO3 ; potassium carbonate

刊名：Bioorganic & Medicinal Chemistry

出版年：2017

5.Inhibitory action of linoleamide and oleamide toward sarco/endoplasmic reticulum Ca²⁺-ATPase

作者：Sachiko Yamamoto^a ; ^{s_yamamoto@ks.kyorin-u.ac.jp} ; Munenori Takehara^b ; Makoto Ushimaru^a

关键词：[Ca2+]cyto ; cytosolic Ca2+ concentration ; ER ; endoplasmic reticulum ; PFAA ; primary fatty acid amide ; SR ; sarcoplasmic reticulum ; SERCA ; sarco/endoplasmic reticulum Ca2+-ATPase ; rSERCA1a ; rabbit SERCA isoform 1a ; hSERCA2b ; human SERCA isoform 2b ; hSERCA3a ; human SERCA isoform 3a

刊名：Biochimica et Biophysica Acta (BBA) - General Subjects

出版年：2017

6.In vitro and in silico studies of the interaction of three tetrazoloquinazoline derivatives with DNA and BSA and their cytotoxicity activities against MCF-7, HT-29 and DPSC cell lines

作者：Maryam Mohamadi^a ; ^{m.mohamadi794@gmail.com} ; Asadollah Hassankhani^b ; S. Yousef Ebrahimipour^c ; Masoud Torkzadeh-Mahani^d

关键词：BSA and DNA interaction ; Molecular docking ; Spectroscopic techniques ; MTT assays ; [123 ; 4]tetrazolo[5 ; 1-b]-quinazolin-8-one derivatives

刊名：International Journal of Biological Macromolecules

出版年：2017

7.Interactions between α-amylase and an acidic branched polysaccharide from green tea

作者：Shuyun Wu ; Minghua Lai ; Jiahao Luo ; Jingwen Pan ; Li-Ming Zhang ; Liqun Yang ; ^{yanglq@mail.sysu.edu.cn}

关键词：Branched acidic tea polysaccharide ; α-amylase ; Interaction

刊名：International Journal of Biological Macromolecules

出版年：2017

8.C0818, a novel curcumin derivative, interacts with Hsp90 and inhibits Hsp90 ATPase activity

作者：Yingjuan Fan^a ; ^b ; Yang Liu^a ; ^b ; Lianru Zhang^c ; Fang Cai^a ; ^b ; Liping Zhu^a ; ^b ; Jianhua Xu^a ; ^b ; ^{xjh@mail.fjmu.edu.cn}

关键词：Curcumin derivative ; Hsp90 ; ATPase activity ; Fluorescence spectrometry ; Interaction

刊名：Acta Pharmaceutica Sinica B

出版年：2017

9.In vitro biopharmaceutical evaluation of ciprofloxacin/metal cation complexes for pulmonary administration

作者：J Brillault^a ; ^b ; ^{julien.brillault@univ-poitiers.fr} ; F Tewes^a ; ^b ; ^{frederic.tewes@univ-poitiers.fr} ; W Couet^a ; ^b ; ^c ; ^{william.couet@univ-poitiers.fr} ; JC Olivier^a ; ^b ; ^{jean.christophe.olivier@univ-poitiers.fr}

关键词：Ciprofloxacin (PubChem CID ; 2764)

刊名：European Journal of Pharmaceutical Sciences

出版年：2017

10.Aluminium sulfate exposure: A set of effects on hydrolases from brain, muscle and digestive tract of juvenile Nile tilapia (Oreochromis niloticus)

作者：Vagne Melo Oliveira^a ; Caio Rodrigo Dias Assis^a ; ^{caiodias2@hotmail.com} ; Helane Maria Silva Costa^a ; Raquel Pereira Freitas Silva^b ; Juliana Ferreira Santos^a ; ^b ; Luiz Bezerra Carvalho Jr^a ; Ranilson Souza Bezerra^a ; ^{ransoube@uol.com.br}

关键词：Aluminium ; Biomarker ; Cholinesterase ; Digestive enzyme ; Pixel optical densitometry

刊名：Comparative Biochemistry and Physiology Part C: Toxicology & Pharmacology

出版年：2017

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