均三唑并噻二唑:重要的潜在药物结构单元

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英文篇名：s-Triazolothiadiazoles: A Class of Important Structural Unit for Potential Drugs 作者：肖立伟 ; 肖树强 ; 李政 ; 景学敏 ; 戴富才 英文作者：Xiao Liwei;Xiao Shuqiang;Li Zheng;Jing Xuemin;Dai Fucai;Faculty of Chemistry and Material Science,Langfang Normal University;Traditional Chinese Medicine Rehabilition Division,Dingzhou Peoples Hospital; 关键词：均三唑并噻二唑 ; 生物活性 ; 构效关系 英文关键词：s-Triazolothiadiazoles;;Biological activities;;Structure activity relationship 中文刊名：HXTB 英文刊名：Chemistry 机构：廊坊师范学院化学与材料科学学院;定州市人民医院中医康复科; 出版日期：2019-01-30 出版单位：化学通报 年：2019 期：v.82 基金：河北省教育厅项目(ZD2016046)资助 语种：中文; 页：HXTB201902004 页数：8 CN：02 ISSN：11-1804/O6 分类号：27-34

摘要

均三唑并噻二唑是一类重要的稠杂环化合物,其衍生物具有抗菌、消炎、抗肿瘤、抗结核、酶抑制作用、调节植物生长等多种生物活性。本文按照均三唑并噻二唑类化合物呈现的不同生物活性进行分类,综述了近年来该类化合物在上述领域的研究进展。
        s-Triazolothiadiazoles compounds are a kind of important fused heterocyclic compounds,which have extensive biological activity such as anti-bacterial, anti-inflammatory, anti-tumor, anti-tuberculosis, enzyme inhibition,regulating plant growth activity and so on. According to the different biological activities of striazolothiadiazoles compounds,the research progress of biological activities for the titled compounds in recent years are reviewed.

引文

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