Cu-Catalyzed Direct Amidation of Aromatic C鈥揌 Bonds: An Access to Arylamines

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• 作者：Hui Xu ; Xixue Qiao ; Shiping Yang ; Zengming Shen
• 刊名：Journal of Organic Chemistry
• 出版年：2014
• 出版时间：May 16, 2014
• 年：2014
• 卷：79
• 期：10
• 页码：4414-4422
• 全文大小：462K
• 年卷期：v.79,no.10(May 16, 2014)
• ISSN：1520-6904

文摘

A Cu-catalyzed aromatic C鈥揌 amidation with phthalimide under oxygen as a terminal oxidant without using additional additives has been achieved. This reaction has the broad substrate scope and shows moderate to good yields in most cases. This method is complementary to the previously reported metal-catalyzed C鈥揌 amination systems.